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CAS 1403254-99-8 Tazemetostat (EPZ-6438) molecular structure lightbox
CAS RN: 1403254-99-8

Tazemetostat (EPZ-6438)

Product Availability

Choose a grade to view its available package options.

13 package records12 with current stock3 grade groups
Batch No.PackageAvailabilityWarehouseLead TimeInquiry
Batchno.20251229 100mg In stock Shanghai Inquiry
Batchno.20251008 1g In stock Shanghai, Shenzhen, Tianjin, Chengdu Inquiry
Batchno.20260603 1mg In stock Shanghai Inquiry
Batchno.20260312 250mg In stock Shanghai, Shenzhen, Wuhan Inquiry
Batchno.20260121 50mg In stock Shanghai, Tianjin Inquiry
Batchno.20260116 5g In stock Shanghai, Shenzhen Inquiry
Batchno.20250512 5mg In stock Shanghai Inquiry
Batch No.PackageAvailabilityWarehouseLead TimeInquiry
Batchno.20260114 100mg In stock Shanghai, Shandong, Chongqing Inquiry
Batchno.20250316 1g In stock Shanghai, Shandong, Guangdong Inquiry
Batchno.20250206 25mg In stock Shanghai, Shandong, Hebei Inquiry
Batchno.20250211 5g Out of stock 5-7 business days Inquiry
Batchno.20251013 5mg In stock Shandong, Guangdong Inquiry
Batch No.PackageAvailabilityWarehouseLead TimeInquiry
Batchno.20251110 1ml In stock Inquiry
  • Product code: SSC-050875
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Verified Factory Data

Supply Overview & Packaging Options

Packaging options, recorded purity, stock quantity and ship-from location below are generated from the current factory data table for this CAS.

  • Pack sizes on record: 0.1g, 0.25g, 1g, 5g
  • Available purity: >97%
  • Inventory rows with stock: 3
  • Bulk packaging: confirmed by inquiry
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Available Pack Sizes & Stock

Specific stock quantities are shown below. Price is not displayed online and is confirmed by inquiry.

Recorded sizes, purity and stock details for CAS 1403254-99-8
Pack Size Recorded Purity Available Qty Ship From Inquiry
0.1g >97% 1 In Stock Hong Kong Inquiry
0.25g >97% 1 In Stock Hong Kong Inquiry
1g >97% 1 In Stock Hong Kong Inquiry
5g >97% 0 Out of Stock Beijing Inquiry

1403254-99-8 / N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-[ethyl(oxan-4-yl)amino]-2-methyl-5-[4-(morpholin-4-ylmethyl)phenyl]benzamide

Standard CAS: 1403254-99-8 Multi CAS: No
Basic Information Computed Properties

Basic Information

CAS
1403254-99-8
Multi CAS
No
Molecular Formula
C34H44N4O4
Molecular Weight
572.700000
Exact Mass
572.336256
SMILES
CCN(C1CCOCC1)C2=CC(=CC(=C2C)C(=O)NCC3=C(C=C(NC3=O)C)C)C4=CC=C(C=C4)CN5CCOCC5
InChI
InChI=1S/C34H44N4O4/c1-5-38(29-10-14-41-15-11-29)32-20-28(27-8-6-26(7-9-27)22-37-12-16-42-17-13-37)19-30(25(32)4)33(39)35-21-31-23(2)18-24(3)36-34(31)40/h6-9,18-20,29H,5,10-17,21-22H2,1-4H3,(H,35,39)(H,36,40)
InChIKey
NSQSAUGJQHDYNO-UHFFFAOYSA-N

Computed Properties

Structural Parameters

Heavy atom count
42
Aromatic heavy atom count
18
Fraction Csp3
0.47
Rotatable bonds
9
H-bond acceptors
6
H-bond donors
2
Molar refractivity
167.28
TPSA
86.9

LogP / Solubility

WLOGP
4.73
MLOGP
4.21
XLogP3
4.2
Consensus LogP
4.38
Log S (ESOL)
-6.1
Class (ESOL)
Insoluble
Log S (Ali)
-7.67
Class (Ali)
Insoluble
Log S (SILICOS-IT)
-8.39
Class (SILICOS-IT)
Insoluble

ADME

GI absorption
High
BBB permeant
No
P-gp substrate
No
CYP1A2 inhibitor
No
CYP2C19 inhibitor
Yes
CYP2C9 inhibitor
No
CYP2D6 inhibitor
Yes
CYP3A4 inhibitor
Yes
Log Kp (skin permeation)
-2.85

Drug-likeness / Medicinal Chemistry

Lipinski
Yes
Ghose
No
Veber
Yes
Egan
Yes
Muegge
Yes
Bioavailability score
0.55
Leadlikeness
No
Synthetic Accessibility
5

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